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Al-Azhar University – Gaza
2009
Biological and Pharmaceutical Bulletin
Docking simulations and in vitro assay unveil potent inhibitory action of papaverine against protein tyrosine phosphatase 1B
32
4
640
645
Faculty of Pharmacy, University of Jordan, Amman 11942, Jordan; Faculty of Pharmacy, Applied Science Private University, Amman, Jordan; Faculty of Pharmacy, Al-Azhar University, Gaza, Gaza Strip, Palestine
21
10.1248/bpb.32.640
Animals; Blood Glucose; Computer Simulation; Dose-Response Relationship, Drug; Humans; Male; Mice; Mice, Inbred BALB C; Models, Molecular; Papaverine; Phosphodiesterase Inhibitors; Protein Tyrosine Phosphatase, Non-Receptor Type 1; Software; berberine; enzyme inhibitor; glucose; papaverine; protein tyrosine phosphatase 1B; recombinant enzyme; rk 682; unclassified drug; animal experiment; article; computer simulation; concentration response; controlled study; diet restriction; dose response; drug activity; drug conformation; drug dose comparison; drug dose escalation; drug effect; drug formulation; drug potency; drug protein binding; drug stability; drug structure; energy; enzyme inhibition; glucose blood level; hydrophobicity; hypoglycemic activity; IC 50; in vitro study; in vivo study; ionization; male; molecular docking; molecular interaction; mouse; nonhuman