Skip to header Skip to main navigation Skip to main content Skip to footer
Home
Academic Citations from Palestine
Foregrounding the Research of Academics in Palestine

Main navigation

  • Home
  • Search
  • About

Synthesis and in vitro evaluation of thiadiazole derivatives as AChE, Bu-ChE and LOX inhibitors

Blank
Al-Azhar University – Gaza
Altintop M.D.; Özdemir A.; Abu Mohsen U.; Temel H.E.; Akal G.; Kaplancikli Z.A.
Altintop, Mehlika Dilek (38662171400); Özdemir, Ahmet (7006505091); Abu Mohsen, Usama (6505829502); Temel, Halide Edip (16231520900); Akal, Gülşen (60208437500); Kaplancikli, Zafer Asim (6602311259)
38662171400; 7006505091; 6505829502; 16231520900; 60208437500; 6602311259
2014
Letters in Drug Design and Discovery
Synthesis and in vitro evaluation of thiadiazole derivatives as AChE, Bu-ChE and LOX inhibitors
11
9
1062
1069
Bentham Science Publishers B.V.
Anadolu University, Faculty of Pharmacy, Department of Pharmaceutical Chemistry, Eskişehir, 26470, Turkey; Al-Azhar University, Faculty of Pharmacy, Department of Pharmaceutical Chemistry, Gaza, Palestine; Anadolu University, Faculty of Pharmacy, Department of Biochemistry, Eskişehir, 26470, Turkey
Altintop M.D., Anadolu University, Faculty of Pharmacy, Department of Pharmaceutical Chemistry, Eskişehir, 26470, Turkey; Özdemir A., Anadolu University, Faculty of Pharmacy, Department of Pharmaceutical Chemistry, Eskişehir, 26470, Turkey; Abu Mohsen U., Al-Azhar University, Faculty of Pharmacy, Department of Pharmaceutical Chemistry, Gaza, Palestine; Temel H.E., Anadolu University, Faculty of Pharmacy, Department of Biochemistry, Eskişehir, 26470, Turkey; Akal G., Anadolu University, Faculty of Pharmacy, Department of Biochemistry, Eskişehir, 26470, Turkey; Kaplancikli Z.A., Anadolu University, Faculty of Pharmacy, Department of Pharmaceutical Chemistry, Eskişehir, 26470, Turkey
A. Özdemir; Anadolu University, Faculty of Pharmacy, Department of Pharmaceutical Chemistry, Eskişehir, 26470, Turkey; email: ahmeto@anadolu.edu.tr
5
10.2174/1570180811666140529004517
Acetylcholinesterase; Butyrylcholinesterase; Lipoxygenase; Thiadiazole.
cholecystokinin octapeptide; cholinesterase inhibitor; lipoxygenase inhibitor; n (3 methoxybenzylidene) 2 [[5 (phenylamino) 1,3,4 thiadiazol 2 yl]thio]acetohydrazide; n' (2 bromobenzylidene) 2 [[5 (phenylamino) 1,3,4 thiadiazol 2 yl]thio]acetohydrazide; n' (2 chlorobenzylidene) 2 [[5 (phenylamino) 1,3,4 thiadiazol 2 yl]thio]acetohydrazide; n' (2 fluorobenzylidene) 2 [[5 (phenylamino) 1,3,4 thiadiazol 2 yl]thio]acetohydrazide; n' (2 methoxybenzylidene) 2 [[5 (phenylamino) 1,3,4 thiadiazol 2 yl]thio]acetohydrazide; n' (2 methylbenzylidene) 2 [[5 (phenylamino) 1,3,4 thiadiazol 2 yl]thio]acetohydrazide; n' (3 bromobenzylidene) 2 [[5 (phenylamino) 1,3,4 thiadiazol 2 yl]thio]acetohydrazide; n' (3 chlorobenzylidene) 2 [[5 (phenylamino) 1,3,4 thiadiazol 2 yl]thio]acetohydrazide; n' (3 fluorobenzylidene) 2 [[5 (phenylamino) 1,3,4 thiadiazol 2 yl]thio]acetohydrazide; n' (3 fuorobenzylidene) 2 [[5 (phenylamino) 1,3,4 thiadiazol 2 yl]thio]acetohydrazide; n' (3 methoxybenzylidene) 2 [[5 (phenylamino) 1,3,4 thiadiazol 2 yl]thio]acetohydrazide; n' (3 methylbenzylidene) 2 [[5 (phenylamino) 1,3,4 thiadiazol 2 yl]thio]acetohydrazide; n' (4 bromobenzylidene) 2 [[5 (phenylamino) 1,3,4 thiadiazol 2 yl]thio]acetohydrazide; n' (4 chlorobenzylidene) 2 [[5 (phenylamino) 1,3,4 thiadiazol 2 yl]thio]acetohydrazide; n' (4 fluorobenzylidene) 2 [[5 (phenylamino) 1,3,4 thiadiazol 2 yl]thio]acetohydrazide; n' (4 methoxybenzylidene) 2 [[5 (phenylamino) 1,3,4 thiadiazol 2 yl]thio]acetohydrazide; n' (4 methylbenzylidene) 2 [[5 (phenylamino) 1,3,4 thiadiazol 2 yl]thio]acetohydazide; n' benzylidene 2 [[5 (phenylamino) 1,3,4 thiadiazol 2yl]thio]acetohydrazide; thiadiazole derivative; unclassified drug; animal cell; Article; drug cytotoxicity; drug synthesis; enzyme assay; enzyme inhibition; human; in vitro study; mouse; nonhuman; physical chemistry; priority journal